1. Signaling Pathways
  2. Antibody-drug Conjugate/ADC Related
  3. Drug-Linker Conjugates for ADC
  4. Drug-Linker Conjugates for ADC Inhibitors

Drug-Linker Conjugates for ADC Inhibitors

Auristatin

Camptothecins

Daunorubicins/Doxorubicins

Duocarmycins

Maytansinoids

Pyrrolobenzodiazepines

Traditional Cytotoxic Agents

Dual payloads

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Drug-Linker Conjugates for ADC Inhibitors & Chemicals
Product Name Auristatin Camptothecins Daunorubicins/Doxorubicins Duocarmycins Maytansinoids Pyrrolobenzodiazepines Traditional Cytotoxic Agents Dual payloads Purity
Deruxtecan  
Camptothecins
            99.94%
VcMMAE
Auristatin
              99.97%
Vipivotide tetraxetan            
Traditional Cytotoxic Agents
  99.46%
Val-Cit-PAB-MMAE
Auristatin
              99.98%
McMMAF
Auristatin
              99.97%
CL2A-SN-38  
Camptothecins
            99.07%
SMCC-DM1        
Maytansinoids
      99.23%
MC-Val-Cit-PAB-MMAF
Auristatin
              98.16%
MC-GGFG-Exatecan  
Camptothecins
            99.71%
DBCO-PEG4-VC-PAB-MMAE      
Duocarmycins
        99.18%
Mal-Gly-PAB-Exatecan-D-glucuronic acid  
Camptothecins
            99.82%
Tesirine          
Pyrrolobenzodiazepines
    98.31%
DBCO-PEG4-GGFG-Dxd            
Traditional Cytotoxic Agents
  98.42%
MC-Val-Cit-PAB-Exatecan  
Camptothecins
            99.57%
MC-VA-PAB-Exatecan  
Camptothecins
            99.58%
AZ14170133  
Camptothecins
            99.73%
Mal-PEG8-Val-Ala-PAB-Exatecan  
Camptothecins
            99.48%
Mc-MMAE
Auristatin
              99.93%
SPDB-DM4        
Maytansinoids
      98.35%
MC-betaglucuronide-MMAE-1
Auristatin
              99.23%
sulfo-SPDB-DM4        
Maytansinoids
      99.97%
Mal-VC-PAB-DM1        
Maytansinoids
      99.41%
DBCO-PEG4-Val-Cit-PAB-MMAF
Auristatin
              98.69%
Gly3-VC-PAB-MMAE
Auristatin
              99.63%
MC-VA-PABC-MMAE
Auristatin
              99.93%
Mal-PEG8-Val-Cit-PAB-MMAE
Auristatin
             
PEG4-aminooxy-MMAF
Auristatin
              99.83%
DBCO-(PEG2-VC-PAB-MMAE)2
Auristatin
           
Dual payloads
99.21%
CL2-SN-38  
Camptothecins
            99.23%
SGD-1910          
Pyrrolobenzodiazepines
   
Vc-seco-DUBA      
Duocarmycins
        99.95%
Gly-Gly-Phe-Gly-NH-O-CO-Exatecan hydrochloride  
Camptothecins
            99.52%
Doxorubicin-SMCC    
Daunorubicins/Doxorubicins
          98.80%
MC-VC-PABC-Aur0101
Auristatin
              99.66%
N3-PEG3-vc-PAB-MMAE
Auristatin
              99.07%
Mal-PEG2-VCP-Eribulin            
Traditional Cytotoxic Agents
  99.82%
SuO-Val-Cit-PAB-MMAE
Auristatin
              99.24%
DM21        
Maytansinoids
      99.92%
DBCO-PEG4-VA-PBD            
Traditional Cytotoxic Agents
  99.68%
Lys-SMCC-DM1        
Maytansinoids
      99.61%
DBCO-PEG4-MMAF
Auristatin
              99.80%
SuO-Glu-Val-Cit-PAB-MMAE
Auristatin
             
MC-Val-Cit-PAB-duocarmycin chloride      
Duocarmycins
        99.04%
MC-Gly-Gly-Phe-Gly-(R)-Cyclopropane-Exatecan  
Camptothecins
           
DBCO-(PEG)3-VC-PAB-MMAE
Auristatin
              99.60%
Mal-PEG2-Gly-Gly-Phe-Gly-Exatecan  
Camptothecins
            99.09%
SC-VC-PAB-MMAE
Auristatin
             
MMAE-SMCC
Auristatin
             
MC-DOXHZN hydrochloride    
Daunorubicins/Doxorubicins
          98.04%
Azide-PEG4-VC-PAB-Doxorubicin    
Daunorubicins/Doxorubicins
          99.62%
Val-Ala-PABC-Exatecan  
Camptothecins
            99.90%
DBCO-PEG3-VC-Exatecan  
Camptothecins
           
Acetylene-linker-Val-Cit-PABC-MMAE
Auristatin
             
Mal-PEG4-VA-PBD          
Pyrrolobenzodiazepines
   
DBM-MMAF
Auristatin
              99.65%
MAC glucuronide phenol-linked SN-38  
Camptothecins
            98.49%
DM4-SMCC        
Maytansinoids
     
Ac-Lys-Val-Cit-PABC-MMAE
Auristatin
              99.94%
P5(PEG24)-VC-PAB-Exatecan  
Camptothecins
            99.74%
Val-Cit-PAB-Exatecan  
Camptothecins
            99.79%
MA-PEG4-VC-PAB-DMEA-duocarmycin DM            
Traditional Cytotoxic Agents
  99.84%
MAL-di-EG-Val-Cit-PAB-MMAE
Auristatin
             
NAMPT inhibitor-linker 2            
Traditional Cytotoxic Agents
  99.35%
MC-Val-Cit-PAB-vinblastine            
Traditional Cytotoxic Agents
 
DBCO-PEG4-VC-PAB-DMEA-PNU-159682      
Duocarmycins
       
2-MSP-5-HA-GGFG-NH-CH2-O-CH2-CO-Exatecan  
Camptothecins
            98.27%
Mal-PEG8-Phe-Lys-PAB-Exatecan TFA  
Camptothecins
            98.44%
AcLys-PABC-VC-Aur0101
Auristatin
              98.49%
Mal-Phe-C4-VC-PAB-MMAE
Auristatin
              99.54%
MC-DM1        
Maytansinoids
      99.50%
CB07-Exatecan  
Camptothecins
            98.97%
PSMA-Val-Cit-PAB-MMAE
Auristatin
              99.52%
PSMA-ALB-56            
Traditional Cytotoxic Agents
  98.92%
GGFG-amide-glycol-amide-Exatecan  
Camptothecins
            98.73%
Fmoc-GGFG-DXd            
Traditional Cytotoxic Agents
  99.81%
Fmoc-Val-Cit-PAB-MMAE
Auristatin
              98.85%
Mal-C6-α-Amanitin    
Daunorubicins/Doxorubicins
          98.48%
Val-Cit-PAB-MMAF sodium
Auristatin
              98.43%
SPP-DM1        
Maytansinoids
     
DBM-GGFG-NH-O-CO-Exatecan  
Camptothecins
           
DBCO-β-Glu-PEG12-Exatecan  
Camptothecins
           
VcMMAE-Deruxtecan              
Dual payloads
98.10%
Mc-MMAD
Auristatin
              98.39%
DM1-PEG4-DBCO        
Maytansinoids
      98.04%
Vc-MMAD
Auristatin
              99.96%
MC-Gly-Gly-Phe-Gly-Cyclobutanecarboxylic-Exatecan  
Camptothecins
            99.55%
NAMPT inhibitor-linker 1            
Traditional Cytotoxic Agents
  99.27%
MC-Gly-Gly-Phe-Gly-GABA-Exatecan  
Camptothecins
            99.72%
Val-Cit-PABC-DOX            
Traditional Cytotoxic Agents
 
GGFG-PAB-MMAE
Auristatin
              99.27%
MC-VC-PABC-C6-α-Amanitin    
Daunorubicins/Doxorubicins
          98.88%
MC-VC-PABC-DNA31            
Traditional Cytotoxic Agents
  98.71%
MC-Val-Cit-PAB-Auristatin E
Auristatin
             
Val-Ala-PABC-Exatecan trifluoroacetate  
Camptothecins
            98.39%
Aminobenzenesulfonic auristatin E TFA
Auristatin
              99.39%
TLR7/8 agonist 4 hydroxy-PEG10-acid hydrochloride            
Traditional Cytotoxic Agents
  98.28%
Cyclooctyne-O-amido-PEG4-VC-PAB-Gly-Gly-NH-O-CO-Exatecan  
Camptothecins
           
BCN-HS-PEG2(vcPABC-MMAE)2              
Dual payloads
(Rac)-Lys-SMCC-DM1        
Maytansinoids
      98.18%
MC-Val-Cit-PAB-carfilzomib iodide            
Traditional Cytotoxic Agents
 
MC-Gly-Gly-Phe-Gly-amide-cyclopropanol-amide-Exatecan  
Camptothecins
            99.16%
Cys-mcMMAD
Auristatin
              98.77%
MC-Val-Cit-PAB-Retapamulin            
Traditional Cytotoxic Agents
  99.00%
MC-Val-Cit-PAB-rifabutin            
Traditional Cytotoxic Agents
 
Fmoc-Val-Cit-PAB-Duocarmycin TM      
Duocarmycins
        99.44%
DBCO-PEG4-Ahx-DM1        
Maytansinoids
     
Lys-Nε-SPDB-DM4        
Maytansinoids
      99.81%
MCC-Modified Daunorubicinol    
Daunorubicins/Doxorubicins
         
MC-Val-Cit-PAB-clindamycin            
Traditional Cytotoxic Agents
  99.99%
MAL-di-EG-Val-Cit-PAB-MMAF
Auristatin
              98.56%
Mal-PEG4-VC-PAB-DMEA-Seco-Duocarmycin SA      
Duocarmycins
       
Aminobenzenesulfonic auristatin E
Auristatin
             
MC-Val-Cit-PAB-Indibulin            
Traditional Cytotoxic Agents
 
MAC glucuronide α-hydroxy lactone-linked SN-38  
Camptothecins
           
MC-GGFG-(7ethanol-10NH2-11F-Camptothecin)  
Camptothecins
           
MA-PEG4-VC-PAB-DMEA-duocarmycin DM TFA            
Traditional Cytotoxic Agents
  99.05%
MC-DOXHZN    
Daunorubicins/Doxorubicins
         
MC-Sq-Cit-PAB-Gefitinib            
Traditional Cytotoxic Agents
 
Sulfo-PDBA-DM4        
Maytansinoids
     
HS-(CH2)3CO-L-Ala-D-Ala-L-Ala-NH-CH2-S-(CH2)5-CO-DM        
Maytansinoids
     
ST8155AA1            
Traditional Cytotoxic Agents
 
MC-Val-Cit-PAB-dimethylDNA31            
Traditional Cytotoxic Agents
  99.97%
Nitro-PDS-Tubulysin M
Auristatin
             
Vat-Cit-PAB-Monomethyl Dolastatin 10
Auristatin
             
VcMMAE-Eribulin              
Dual payloads
VCP-Eribulin            
Traditional Cytotoxic Agents
 
Gly-Mal-Gly-Gly-Phe-Gly-amide-methylcyclopropane-Exatecan  
Camptothecins
           
Val-Cit-PAB-MMAF
Auristatin
             
TLR7/8 agonist 4 hydroxy-PEG10-acid            
Traditional Cytotoxic Agents
 
MC-Gly-Gly-Phe-Gly-(S)-Cyclopropane-Exatecan  
Camptothecins
           
DM4-SPDP        
Maytansinoids
     
Deruxtecan-Eribulin              
Dual payloads
MP-PEG8-Val-Lys-Ala-7-MAD-MDCPT  
Camptothecins
           
DBA-DM4        
Maytansinoids
     
MC-Alkyl-Hydrazine Modified MMAF
Auristatin
             
Mal-cyclohexane-Gly-Gly-Phe-Gly-Exatecan  
Camptothecins
           
Val-Cit-Exatecan TFA            
Traditional Cytotoxic Agents
 
MC-VC-PAB-Tubulysin M
Auristatin
             
MC-VC(S)-PABQ-Tubulysin M
Auristatin
             
Sulfo-SPDB-DGN462        
Maytansinoids
     
Desmethyl Vc-seco-DUBA      
Duocarmycins
       
MC-betaglucuronide-MMAE-2
Auristatin
             
ST8154AA1            
Traditional Cytotoxic Agents
 
Mal-PEG8-Phe-Lys-PAB-Exatecan  
Camptothecins
           
Rha-PEG3-SMCC            
Traditional Cytotoxic Agents
 
MB-VC-MGBA      
Duocarmycins
       
MC-Sq-Cit-PAB-Dolastatin10
Auristatin
             
N3-PEG8-Phe-Lys-PABC-Gefitinib            
Traditional Cytotoxic Agents
 
Aminooxy CatB-LXR            
Traditional Cytotoxic Agents
 
OSu-Glu-VC-PAB-MMAD
Auristatin
             
AMCC-DM1        
Maytansinoids
     
LE01  
Camptothecins
           
Mal-VC-PAB-EDA-N-Ac-Calicheamicin            
Traditional Cytotoxic Agents
 
AcLysValCit-PABC-DMAE-SW-163D            
Traditional Cytotoxic Agents
 
AmPEG6C2-Aur0131            
Traditional Cytotoxic Agents